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Volume 58, Number 2, February 2006

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Review Article

In-vitro and in-vivo assays for angiogenesis-modulating drug discovery and development
pp. 153-160(8)
Authors: Phung, Michelle W.; Dass, Crispin R.

Research Papers: Pharmaceutics and Drug Delivery

Skin permeation of retinol in Tween 20-based deformable liposomes: in-vitro evaluation in human skin and keratinocyte models
pp. 161-166(6)
Authors: Oh, Yu-Kyoung; Kim, Mi Young; Shin, Jee-Young; Kim, Tae Woon; Yun, Mi-Ok; Yang, Sung Joon; Choi, Sang Sook; Jung, Woon-Won; Kim, Jung Ae; Choi, Han-Gon

Design, synthesis and characterization of captopril prodrugs for enhanced percutaneous absorption
pp. 167-177(11)
Authors: Moss, Gary P.; Gullick, Darren R.; Cox, Paul A.; Alexander, Cameron; Ingram, Matthew J.; Smart, John D.; Pugh, W. John

Characterization of pilocarpine-loaded chitosan/Carbopol nanoparticles
pp. 179-186(8)
Authors: Kao, Huei-Jen; Lin, Hong-Ru; Lo, Yu-Li; Yu, Shi-Ping

Amphiphilogels as drug carriers: effects of drug incorporation on the gel and on the active drug
pp. 187-194(8)
Authors: Jibry, Nadeen; Sarwar, Tanzeem; Murdan, Sudaxshina

Research Papers: Biopharmaceutics and Drug Disposition

Activation of P2Y receptor enhances high-molecular compound absorption from rat ileum
pp. 195-200(6)
Authors: Kinoshita, Natsumi; Takahashi, Tomoko; Tada, Shoko; Shinozuka, Kazumasa; Mizuno, Nobuyasu; Takahashi, Koichi

Research Papers: Molecular and Clinical Pharmacology

Synthesis and binding profile of constrained analogues of N-[4-(4-arylpiperazin-1-yl)butyl]-3-methoxybenzamides, a class of potent dopamine D3 receptor ligands
pp. 209-218(10)
Authors: Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola A.; Berardi, Francesco; Perrone, Roberto

Evaluation of in-vitro anti-inflammatory activity of some 2-alkyl-4,6-dimethoxy-1,3,5-triazines
pp. 219-226(8)
Authors: Dianzani, Chiara; Collino, Massimo; Gallicchio, Margherita; Samaritani, Simona; Signore, Giovanni; Menicagli, Rita; Fantozzi, Roberto

Mechanism underlying mitochondrial protection of asiatic acid against hepatotoxicity in mice
pp. 227-233(7)
Authors: Gao, Jing; Chen, Jin; Tang, Xinhui; Pan, Liya; Fang, Feng; Xu, Lizhi; Zhao, Xiaoning; Xu, Qiang

Research Papers: Drugs from Natural Sources

In-vitro and in-vivo antitumour activity of physalins B and D from Physalis angulata
pp. 235-241(7)
Authors: Magalhães, Hemerson Iury Ferreira; Veras, Maria Leopoldina; Torres, Márcia Rocha; Alves, Ana Paula Negreiros Nunes; Pessoa, Otília Deusdênia Loiola; Silveira, Edilberto Rocha; Costa-Lotufo, Letícia Veras; de Moraes, Manoel Odorico; Pessoa, Cláudia

Effects of Ginkgo biloba extract on blood pressure and vascular endothelial response by acetylcholine in spontaneously hypertensive rats
pp. 243-249(7)
Authors: Kubota, Yoko; Tanaka, Naoko; Kagota, Satomi; Nakamura, Kazuki; Kunitomo, Masaru; Umegaki, Keizo; Shinozuka, Kazumasa

In-vitro effect of flavonoids from Solidago canadensis extract on glutathione S-transferase
pp. 251-256(6)
Authors: Apáti, Pál; Houghton, Peter J.; Kite, Geoffrey; Steventon, Glyn B.; Kéry, Ágnes

Protective effect of Nardostachys jatamansi on oxidative injury and cellular abnormalities during doxorubicin-induced cardiac damage in rats
pp. 257-262(6)
Authors: Subashini, Rajakannu; Yogeeta, Surinderkumar; Gnanapragasam, Arunachalam; Devaki, Thiruvengadam

Communications

Paracellular and transcellular pathways facilitate insulin permeability in rat gut
pp. 271-275(5)
Authors: Lane, Majella E.; Corrigan, Owen I.

Protective effects of Swertia longifolia Boiss. and its active compound, swerchirin, on paracetamol-induced hepatotoxicity in mice
pp. 277-280(4)
Authors: Hajimehdipoor, Homa; Sadeghi, Zhina; Elmi, Sara; Elmi, Azadeh; Ghazi-Khansari, Mahmoud; Amanzadeh, Yaghoub; Sadat-Ebrahimi, Seyyed-Esmaeal

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